The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 27589480 |
72 |
Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH |
Takeda Pharmaceutical |
| 25811530 |
20 |
Rational design of triazololipopeptides analogs of kisspeptin inducing a long-lasting increase of gonadotropins. |
Umr7247 |
| 24918545 |
81 |
Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity. |
Takeda Pharmaceutical |
| 24047141 |
64 |
Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity. |
Takeda Pharmaceutical |
| 22995619 |
22 |
Trypsin resistance of a decapeptide KISS1R agonist containing an N¿-methylarginine substitution. |
Takeda Pharmaceutical |
| 22975302 |
45 |
Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides. |
Takeda Pharmaceutical |
| 24900254 |
14 |
Activation of Neuropeptide FF Receptors by Kisspeptin Receptor Ligands. |
TBA |
| 20580563 |
42 |
2-acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats. |
Takeda Pharmaceutical |
| 20457527 |
42 |
Synthesis and structure-activity relationships of 2-acylamino-4,6-diphenylpyridine derivatives as novel antagonists of GPR54. |
Takeda Pharmaceutical |
| 17579384 |
27 |
SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54. |
Kyoto University |
| 17266198 |
84 |
Metastin (KiSS-1) mimetics identified from peptide structure-activity relationship-derived pharmacophores and directed small molecule database screening. |
University of Minnesota Health Science Center |
| 30598349 |
30 |
A new class of pentapeptide KISS1 receptor agonists with hypothalamic-pituitary-gonadal axis activation. |
Takeda Pharmaceutical |
| 19007202 |
12 |
Development of Novel G-Protein-Coupled Receptor 54 Agonists with Resistance to Degradation by Matrix Metalloproteinase. |
Kyoto University |
Search and Browse
